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Mutations in rv0678 confer low-level resistance to benzothiazinone DprE1 inhibitors in M. tuberculosis

ACLY inhibitors induce apoptosis and potentiate cytotoxic effects of sorafenib in thyroid cancer cells

JoF, Vol. 8, Pages 688: Triazole Derivatives Target 14α–Demethylase (LDM) Enzyme in Candida albicans Causing Ergosterol Biosynthesis Inhibition

CIMB, Vol. 44, Pages 2825-2841: Identification of Putative Plant-Based ALR-2 Inhibitors to Treat Diabetic Peripheral Neuropathy

Inhibitors of ROCK kinases induce multiple mitotic defects and synthetic lethality in BRCA2-deficient cells

Pharmaceuticals, Vol. 15, Pages 799: Design, Synthesis and Molecular Docking of Novel Acetophenone-1,2,3-Triazoles Containing Compounds as Potent Enoyl-Acyl Carrier Protein Reductase (InhA) Inhibitors

Viruses, Vol. 14, Pages 1404: Inhibitors of Deubiquitinating Enzymes Interfere with the SARS-CoV-2 Papain-like Protease and Block Virus Replication In Vitro

Cancers, Vol. 14, Pages 3153: 3-Bromo-Isoxazoline Derivatives Inhibit GAPDH Enzyme in PDAC Cells Triggering Autophagy and Apoptotic Cell Death

Bioluminescence-based reporters for characterizing inhibitors and activators of human Sonic Hedgehog protein autoprocessing in live cells at high throughput.

Broadening the Scope of Biocatalysis Engineering by Tailoring Enzyme Microenvironment: A Review

Renin–Angiotensin–Aldosterone Inhibitors and COVID-19 Infection

DYRK1A inhibitors and perspectives for the treatment of Alzheimer's disease

Mechanistic Analysis of Chemically Diverse Bromodomain-4 Inhibitors Using Balanced QSAR Analysis and Supported by X-ray Resolved Crystal Structures

Study of the dynamic behavior of the cruzain enzyme in free and complexed forms with competitive and noncovalent benzimidazole inhibitors

An in silico molecular modeling approach of halolactone derivatives as potential inhibitors for human immunodeficiency virus type-1 reverse transcriptase enzyme

Identification of novel small molecule inhibitors for endoplasmic reticulum oxidoreductase 1α (ERO1α) enzyme: structure-based molecular docking and molecular dynamic simulation studies

Synthesis of new urease enzyme inhibitors as antiulcer drug and computational study

Unraveling the potential role of bioactive molecules produced by Trichoderma spp. as inhibitors of tomatinase enzyme having an important role in wilting disease: an in-silico approach

Potential inhibitors of angiotensin converting enzyme 2 receptor of COVID-19 by Corchorus olitorius Linn using docking, molecular dynamics, conceptual DFT investigation and pharmacophore mapping

In silico design of enzymeα-amylase and α-glucosidase inhibitors using molecular docking, molecular dynamic, conceptual DFT investigation and pharmacophore modelling

Kidney Angiotensin in Cardiovascular Disease: Formation and Drug Targeting [Review Article]

A dual-target herbicidal inhibitor of lysine biosynthesis

Inhibitors of catechol-O-methyltransferase sensitize mice to pain.

Inhibitors of catechol-O-methyltransferase sensitize mice to pain.

Inhibitors of catechol-O-methyltransferase sensitize mice to pain.

Inhibitors of a Na+-pumping NADH-ubiquinone oxidoreductase play multiple roles to block enzyme function [Enzymology]

Inhibitors of catechol-O-methyltransferase sensitize mice to pain

Inhibitors of Human 5-Lipoxygenase Potently Interfere With Prostaglandin Transport

Inhibitors of Advanced Glycation End Product (AGE) Formation and Accumulation.

Enzyme Inhibitory Kinetics and Molecular Docking Studies of Halo-Substituted Mixed Ester/Amide-Based Derivatives as Jack Bean Urease Inhibitors

Enzyme Inhibitory Kinetics and Molecular Docking Studies of Halo-Substituted Mixed Ester/Amide-Based Derivatives as Jack Bean Urease Inhibitors

Mathematical expressions describing enzyme velocity and inhibition at high enzyme concentration

Mechanistic cross-talk between DNA/RNA polymerase enzyme kinetics and nucleotide substrate availability in cells: Implications for polymerase inhibitor discovery [Metabolism]

Environmental and biomedical applications of enzyme inhibitors

Antibiotics, Vol. 9, Pages 595: Indoline-6-Sulfonamide Inhibitors of the Bacterial Enzyme DapE

Renin inhibitors versus angiotensin converting enzyme (ACE) inhibitors for primary hypertension.

Renin inhibitors versus angiotensin converting enzyme (ACE) inhibitors for primary hypertension.

Comparison of the active sites of DNMT2 and COMT and virtual screening for finding new inhibitors

Inhibition of Cytochrome P450 Enzyme and Drug‑Drug Interaction Potential of Acid Reducing Agents Used in Management of CDK inhibitors for Breast Cancer Chemotherapy

Design, synthesis and biological assessment of new selective COX-2 inhibitors including methyl sulfonyl moiety.

Aptamer-functionalized magnetic nanoparticles conjugated organic framework for immobilization of acetylcholinesterase and its application in inhibitors screening.

Diverse chemical space of indoleamine-2,3-dioxygenase 1 (Ido1) inhibitors.

New potent and selective cytochrome P450 2B6 (CYP2B6) inhibitors based on three-dimensional quantitative structure-activity relationship (3D-QSAR) analysis.

Identification of inhibitors of the nicotine metabolising CYP2A6 enzyme-an in silico approach.

Differing Effects of Two Angiotensin Converting Enzyme Inhibitors, Captopril and CI-906, on Diuresis and the Urinary Excretion of Kallikrein and Prostaglandins in Spontaneously Hypertensive Rats.

Differing Effects of Two Angiotensin Converting Enzyme Inhibitors, Captopril and CI-906, on Diuresis and the Urinary Excretion of Kallikrein and Prostaglandins in Spontaneously Hypertensive Rats.

Differing Effects of Two Angiotensin Converting Enzyme Inhibitors, Captopril and CI-906, on Diuresis and the Urinary Excretion of Kallikrein and Prostaglandins in Spontaneously Hypertensive Rats.

Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents.

Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors.